(73) Lexicon Pharmaceuticals, Inc., The Woodlands, TX 77381, 8800 Technology
Forest Place (US)
(54) IMIDAZOLBASIERTE VERBINDUNGEN, ZUSAMMENSETZUNGEN DAMIT
UND VERFAHREN ZU IHRER ANWENDUNG
(72) AUGERI, David, J., Princeton, NJ 08540, 107 Carter Road (US)
(72) BAGDANOFF, Jeffrey, Robbinsville, NJ 08691, 31 Beacon Court (US)
(72) BOTEJU, Lakmal, W., Kendall Park, NJ 08824, 5 Brittany Way (US)
(72) CARSON, Kenneth, G., Princeton, NJ 08540, 96 Herrontown Road (US)
(72) JESSOP, Theodore, C., Lawrenceville, NJ 08648, 31 Merion Place (US)
(72) KIMBALL, David, S., East Winsor, NJ 08520, 13 Charred Oak Lane (US)
(30) US 2006 02 24 776473 P
(30) US 2006 06 20 815221 P
(30) US 2007 01 25 698253
(73) Probiodrug AG, 06120 Halle/Saale, Weinbergweg 22 (DE)
(54) CYANOGUANIDINDERIVATE ALS INHIBITOREN VON
GLUTAMINYLCYCLASE
(72) BUCHHOLZ, Mirko, 06114 Halle/Saale, Brandenburger Strasse 6 (DE)
(72) HEISER, Ulrich, 06108 Halle/Saale, Franz-Schubert-Strasse 5 (DE)
(72) HOFFMANN, Torsten, 06114 Halle/Saale, Koernerstrasse 8 (DE)
(72) BÖHME, Livia, 06126 Halle/Saale, Falterweg 6a (DE)
(30) US 2007 04 18 912528 P
(73) CIPLA LIMITED, Mumbai 400 008, Mumbai Central (IN)
(54) VERFAHREN FÜR DIE ZUBEREITUNG VON LEVOSIMENDAN UND
ZWISCHENPRODUKTE ZUR VERWENDUNG IN DEM VERFAHREN
(72) RAO, Dharmaraj, Ramachandra, Maharashtra, 4/403, Garden Enclave
Pokhran Road 2 Thane (W) 400 601 (IN)
(72) KANKAN, Rajendra, Narayanrao, Maharashtra, 1204 Heritage
HiranandaniGardens Powai Mumbai 400 076 (IN)
(72) PHULL, Manjinder, Singh, Maharashtra, Gobind Niwas Bhattipada Road
Bhandup Mumbai 400 078 (IN)
(72) SAWANT, Ashwini, Amol, Maharashtra, B-605 Akruti Elegance Gavapada
Mulund (East) Mumbai 400 081 (IN)
(30) IN 2009 07 14 MU16452009
(73) BASF SE, 67056 Ludwigshafen (DE)
(54) VERFAHREN ZUR HERSTELLUNG VON 3-PHENYL(THIO)URACILEN UND
- DITHIOURACILEN
(72) LÖHR, Sandra, 67059 Ludwigshafen, Benckiser Str. 30 (DE)
(72) GEBHARDT, Joachim, 67157 Wachenheim, Pegauer Str. 51 (DE)
(72) MAYER, Guido, 67161 Gönnheim, Paul-Münch-Weg 7 (DE)
(72) KEIL, Michael, 67251 Freinsheim, Fontanestr.4 (DE)
(72) SCHMIDT, Thomas, 67433 Neustadt, Pfarrgasse 8 (DE)
(72) WOLF, Bernd, 67136 Fussgönheim, Halbergstr. 4 (DE)
(30) DE 2004 07 22 102004035656
(73) Symphony Evolution, Inc., Rockville, MD 20850, 7361 Calhoun Place, Suite
325 (US)
(54) Verfahren zur Herstellung von Rezeptorkinase-Modulatoren
(72) Rice, Kenneth D., San Rafael, CA 94903, 444 Montecillo Road (US)
(72) Anand, Neel Kumar, San Mateo, CA 94403, 2713 South Norfolk Street Apt.
No. 206 (US)
(72) Bussenius, Joerg, Foster City, CA 94404, 1042 Ilem Lane (US)
(72) Costanza, Simona, Atherton, CA 94027, 51, Jennings Lane (US)
(72) Kennedy, Abigail R., Oakland, CA 94601, 2417 East 28th Street (US)
(72) Kim, Angie I., San Mateo, CA 94404, 928 Shoal Drive (US)
(72) Peto, Csaba J., Alameda, CA 94501, 965 Shorepoint Court, No. 305 (US)
(72) Tsang, Tsze H., El Cerrito, CA 94530, 8367 Kent Drive (US)
(72) Blazey, Charles M., San Francisco, CA 94118, 201 Cornwall Street, No. 3
(US)
(30) US 2002 07 15 396269 P
(30) US 2003 02 13 447212 P
(73) Astellas Pharma Inc., Chuo-ku Tokyo, 3-11, Nihonbashi-Honcho 2-chome (JP)
(72) KONTANI, Toru c/o Astellas Pharma Inc., Chuo-ku, Tokyo 103-8411, 3-11,
Nihonbashi-honcho 2-chome (JP)
(72) MIYATA, Junji c/o Astellas Pharma Inc., Chuo-ku, Tokyo 103-8411, 3-11,
Nihonbashi-honcho 2-chome (JP)
(72) HAMAGUCHI, Wataru c/o Astellas Pharma Inc., Chuo-ku, Tokyo 103-8411, 3-
11, Nihonbashi-honcho 2-chome (JP)
(72) KAWANO, Tomoaki c/o Astellas Pharma Inc., Chuo-ku, Tokyo 103-8411, 3-
11, Nihonbashi-honcho 2-chome (JP)
(72) KAMIKAWA, Akio c/o Astellas Pharma Inc., Chuo-ku, Tokyo 103-8411, 3-11,
Nihonbashi-honcho 2-chome (JP)
(72) SUZUKI, Hiroshi c/o Astellas Pharma Inc., Chuo-ku, Tokyo 103-8411, 3-11,
Nihonbashi-honcho 2-chome (JP)
(72) SUDO, Kenji c/o Astellas Pharma Inc., Chuo-ku, Tokyo 103-8411, 3-11,
Nihonbashi-honcho 2-chome (JP)
(30) JP 2003 08 08 2003290850
(73) Taisho Pharmaceutical Co., Ltd., Tokyo 170-8633, 24-1, Takada 3-chome
Toshima-ku (JP)
(72) ONO, Naoya, Toshima-ku, Tokyo 170-8633, Taisho Pharmaceutical Co., Ltd.
24-1, Takada 3-chome (JP)
(72) TAKAYAMA, Tetsuo, Toshima-ku, Tokyo 170-8633, Taisho Pharmaceutical
Co., Ltd. 24-1, Takada 3-chome (JP)
(72) SHIOZAWA, Fumiyasu, Toshima-ku, Tokyo 170-8633, Taisho Pharmaceutical
Co., Ltd. 24-1, Takada 3-chome (JP)
(72) KATAKAI, Hironori, Toshima-ku, Tokyo 170-8633, Taisho Pharmaceutical
Co., Ltd. 24-1, Takada 3-chome (JP)
(72) YABUUCHI, Tetsuya, Toshima-ku, Tokyo 170-8633, Taisho Pharmaceutical
Co., Ltd. 24-1, Takada 3-chome (JP)
(72) OTA, Tomomi, Toshima-ku, Tokyo 170-8633, Taisho Pharmaceutical Co., Ltd.
24-1, Takada 3-chome (JP)
(72) YAGI, Makoto, Toshima-ku, Tokyo 170-8633, Taisho Pharmaceutical Co., Ltd.
24-1, Takada 3-chome (JP)
(72) SATO, Masakazu, Toshima-ku, Tokyo 170-8633, Taisho Pharmaceutical Co.,
Ltd. 24-1, Takada 3-chome (JP)
(30) JP 2006 02 03 2006027799
(73) Shionogi & Co., Ltd., Osaka 541-0045, 1-8, Doshomachi 3-chome Chuo-ku
Osaka-shi (JP)
(54) TRIAZINDERIVATE ALS P2X3 UND/ODER P2X2/3 REZEPTOR
ANTAGONISTEN UND PHARMAZEUTISCHE ZUSAMMENSETZUNG, DIE DIESE
ENTHÄLT
(72) KAI, Hiroyuki, Osaka-shi Osaka 553-0002, c/o Shionogi&Co. Ltd. 12-4 Sagisu
5-chome Fukushima-ku (JP)
(72) KAMEYAMA, Takayuki, Koka-shi Shiga 520-3423, c/o Shionogi&Co. Ltd.
1405 Gotanda Kokacho (JP)
(72) HASEGAWA, Tsuyoshi, Osaka-shi Osaka 553-0002, c/o Shionogi&Co. Ltd.
12-4 Sagisu 5-chome Fukushima-ku (JP)
(72) OOHARA, Miho, Osaka-shi Osaka 553-0002, c/o Shionogi&Co. Ltd. 12-4
Sagisu 5-chome Fukushima-ku (JP)
(72) TADA, Yukio, Osaka-shi Osaka 553-0002, c/o Shionogi&Co. Ltd. 12-4 Sagisu
5-chome Fukushima-ku (JP)
(72) ENDOH, Takeshi, Osaka-shi Osaka 553-0002, c/o Shionogi&Co. Ltd. 12-4
Sagisu 5-chome Fukushima-ku (JP)
(30) JP 2009 02 13 2009031520
(30) JP 2009 11 25 2009266903
(73) BASF SE, 67056 Ludwigshafen (DE)
(54) VERFAHREN ZUR HERSTELLUNG 5,5-DISUBSTITUIERTER 4,5-
DIHYDROISOXAZOL-3-THIOCARBOXAMIDIN-SALZE
(72) FRASSETTO, Timo, 68165 Mannheim, Bassermannstrasse 35 (DE)
(73) F.I.S.- Fabbrica Italiana Sintetici S.p.A., 36041 Alte di Montecchio Maggiore
(VI), Viale Milano, 26 (IT)
(54) Verfahren zur Herstellung von Efavirenz
(72) LEGANZA, Alessandro, I-36075 Alte di Montecchio Maggiore (Vicenza), F.I.S.
Fabbrica Italiana Sintetici S.p.A, Viale Milano, 26 (IT)
(72) GALVAGNI, Marco, I-36075 Alte di Montecchio Maggiore (Vicenza), F.I.S.
Fabbrica Italiana Sintetici S.p.A, Viale Milano, 26 (IT)
(73) E. I. du Pont de Nemours and Company, Wilmington, DE 19898, 1007 Market
Street (US)
(54) HYDRIERUNGSVERFAHREN ZUR HERSTELLUNG VON
TETRAHYDROFURAN UND ALKYLIERTEN DERIVATEN DAVON
(72) HUTCHENSON, Keith, W., Lincoln University Pennsylvania 19352, 311
Belmont Court (US)
(72) SENGUPTA, Sourav, Kumar, Wilmington Delaware 19808, 122 Westgate
Drive (US)
(30) US 2009 04 07 167413 P
(73) University Of The Free State, 9301 Bloemfontein, Department of Chemistry
Nelson Mandela Drive (ZA)
(54) SYNTHESE VON C-3-GEKOPPELTEN BIFLAVONOIDEN UND C-3-
GEKOPPELTE BIFLAVONOID-ANALOGA
(72) VAN DER WESTHUIZEN, Jan Hendrik, 9301 Bloemfontein, 7 Clarens Street
Bayswater (ZA)
(72) BONNET, Susanna Lucia, 9301 Bloemfontein, 235 Paul Kruger Avenue
Universitas (ZA)
(72) ACHILONU, Mathew, 9301 Bloemfontein, SK flat A University of the Free
State Nelson Mandela Avenue (ZA)
(72) SISA, Miroslav, 9301 Bloemfontein, Room 16 President Steyn Complex
University of the Free State Campus Nelson Mandela Avenue (ZA)
(30) ZA 2009 08 19 200905765
Österreichisches Patentblatt 111. Jahrgang Nummer 4, Seite 1176
Comentários a estes Manuais